Research
category
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A Comprehensive Biological and Synthetic Perspective on 2-Deoxy-D-Glucose (2-DG), A Sweet Molecule with Therapeutic and Diagnostic Potentials Article (Web of Science)
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A PER2-Derived Mechanism-Based Bisubstrate Analog for Casein Kinase 1 epsilon Article (Web of Science)
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ACS CHEMICAL NEUROSCIENCE Journal
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ACS COMBINATORIAL SCIENCE Journal
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ACS INFECTIOUS DISEASES Journal
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ACS MEDICINAL CHEMISTRY LETTERS Journal
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ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 48 Book
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Amide Bond Bioisosteres: Strategies, Synthesis, and Successes Article (Web of Science)
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BIOORGANIC & MEDICINAL CHEMISTRY Journal
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BIOORGANIC & MEDICINAL CHEMISTRY LETTERS Journal
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Biochemical and microbiological evaluation of N-aryl urea derivatives against mycobacteria and mycobacterial hydrolases Article (Web of Science)
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Biomimetic Syntheses and Antiproliferative Activities of Racemic, Natural (-), and Unnnatural (+) Glyceollin I Article (Web of Science)
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CETZOLE Analogs as Potent Ferroptosis Inducers and Their Target Identification Using Covalent/Affinity Probes Article (Web of Science)
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CHEMBIOCHEM Journal
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CHEMICAL BIOLOGY & DRUG DESIGN Journal
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CHEMICAL RESEARCH IN TOXICOLOGY Journal
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CURRENT MEDICINAL CHEMISTRY Journal
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DRUG DESIGN DEVELOPMENT AND THERAPY Journal
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DRUG DEVELOPMENT AND INDUSTRIAL PHARMACY Journal
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Design and discovery of silybin analogues as antiproliferative compounds using a ring disjunctive - Based, natural product lead optimization approach Article (Web of Science)
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Development of bisubstrate analog inhibitors of aspartate N-acetyltransferase, a critical brain enzyme Article (Web of Science)
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Differential Induction of Cytoplasmic Vacuolization and Methuosis by Novel 2-Indolyl-Substituted Pyridinylpropenones Article (Web of Science)
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Discovery of Novel Inhibitors of a Critical Brain Enzyme Using a Homology Model and a Deep Convolutional Neural Network Article (Web of Science)
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EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY Journal
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Elucidating structural features of an entirely carbohydrate cancer vaccine construct employing circular dichroism and fluorescent labeling Article (Web of Science)
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First-in-Class Dual Mechanism Ferroptosis-HDAC Inhibitor Hybrids Article (Web of Science)
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Furoxans (Oxadiazole-4N-oxides) with Attenuated Reactivity are Neuroprotective, Cross the Blood Brain Barrier, and Improve Passive Avoidance Memory Article (Web of Science)
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Hypoxia Activated Prodrugs of a 9-Aza-anthrapyrazole Derivative That Has Promising Anticancer Activity Article (Web of Science)
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Immunogenic Sulfated l-Idose Homo Oligosaccharides Elicit Neutralizing Antibody against Native Heparan Sulfate with Biomarker and Therapeutic Possibilities Article (Web of Science)
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Investigation of the Anticancer Potential of 2-alkoxycarbonylallyl Esters Against Metastatic Murine Breast Cancer Line 4T1 Targeting the EGFR: A Combined Molecular Docking, QSAR, and Machine Learning Approach Article (Web of Science)
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JOURNAL OF ETHNOPHARMACOLOGY Journal
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JOURNAL OF MEDICINAL CHEMISTRY Journal
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JOURNAL OF NATURAL PRODUCTS Journal
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JOURNAL OF PHARMACEUTICAL SCIENCES Journal
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MEDCHEMCOMM Journal
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MEDICINAL CHEMISTRY Journal
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MEDICINAL CHEMISTRY RESEARCH Journal
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MEDICINAL RESEARCH REVIEWS Journal
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Mycobacterium tuberculosis CitA activity is modulated by cysteine oxidation and pyruvate binding Article (Web of Science)
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New camphor hybrids: lipophilic enhancement improves antimicrobial efficacy against drug-resistant pathogenic microbes and intestinal worms Article (Web of Science)
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Nicotinic Acid Adenine Dinucleotide Phosphate Analogues Containing Substituted Nicotinic Acid: Effect of Modification on Ca2+ Release Article (Web of Science)
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Nicotinic Acid Adenine Dinucleotide Phosphate Analogues Substituted on the Nicotinic Acid and Adenine Ribosides. Effects on Receptor Mediated Ca2+ Release Article (Web of Science)
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PLANTA MEDICA Journal
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Photochemical Generation of a C5-Uridinyl Radical Article (Web of Science)
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Practical synthesis of a chromene analog for use as a retinoic acid receptor alpha antagonist lead compound Article (Web of Science)
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Rational design of metabolically stable HDAC inhibitors: An overhaul of trifluoromethyl ketones Article (Web of Science)
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SAR and molecular mechanism studies of monoamine oxidase inhibition by selected chalcone analogs Article (Web of Science)
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Small Molecule Inhibitors Targeting the "Undruggable" Survivin: The Past, Present, and Future from a Medicinal Chemist's Perspective Article (Web of Science)
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Structure and Activity of the Thermophilic Tryptophan-6 Halogenase BorH Article (Web of Science)
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Structure-Based Discovery of Selective Histone Deacetylase 8 Degraders with Potent Anticancer Activity Article (Web of Science)
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Sulfation of hesperetin, naringenin and apigenin by the human cytosolic sulfotransferases: a comprehensive analysis Article (Web of Science)
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Syntheses of 2,3-Diarylated 2H-Benzo[e][1,2]Thiazine 1,1-Dioxides and their 3,4-Dihydro Derivatives, and Assessment of their Inhibitory Activity Against MCF-7 Breast Cancer Cells Article (Web of Science)
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Synthesis and Biological Evaluation of Indolyl-Pyridinyl-Propenones Having Either Methuosis or Microtubule Disruption Activity Article (Web of Science)
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Synthesis and Evaluation of Indole-Based Chalcones as Inducers of Methuosis, a Novel Type of Nonapoptotic Cell Death Article (Web of Science)
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Synthesis and Evaluation of PPAR delta Agonists That Promote Osteogenesis in a Human Mesenchymal Stem Cell Culture and in a Mouse Model of Human Osteoporosis Article (Web of Science)
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Synthesis and Identification of a Novel Lead Targeting Survivin Dimerization for Proteasome-Dependent Degradation Article (Web of Science)
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Synthesis and biological evaluation of isomeric methoxy substitutions on anti-cancer indolyl-pyridinyl-propenones: Effects on potency and mode of activity Article (Web of Science)
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Synthesis and in Vitro Characterization of Trehalose-Based Inhibitors of Mycobacterial Trehalose 6-Phosphate Phosphatases Article (Web of Science)
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Systematic Design of Adenosine Analogs as Inhibitors of a Clostridioides difficile-Specific DNA Adenine Methyltransferase Required for Normal Sporulation and Persistence Article (Web of Science)
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Targeting the trehalose utilization pathways of Mycobacterium tuberculosis Review Article (Web of Science)
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The Impact of Structure on Oxidatively Generated DNA Damage Products Resulting from the C3 '-Thymidinyl Radical Article (Web of Science)
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The Mycobacterium tuberculosis mycothiol S-transferase is divalent metal-dependent for mycothiol binding and transfer Article (Web of Science)
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Therapeutic Activity of the Lansoprazole Metabolite 5-Hydroxy Lansoprazole Sulfide in Triple-Negative Breast Cancer by Inhibiting the Enoyl Reductase of Fatty Acid Synthase Article (Web of Science)
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Thienopyrimidine derivatives exert their anticancer efficacy via apoptosis induction, oxidative stress and mitotic catastrophe Article (Web of Science)
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Tunable Cysteine-Targeting Electrophilic Heteroaromatic Warheads Induce Ferroptosis Article (Web of Science)